Property Name |
Property Value |
Unit |
Raw Value |
Raw Unit |
Annotation |
Reference |
Bioavailability |
58.0 |
% |
58 |
% |
PO, oral; |
DRUGBANK |
T Max |
1.0 |
h |
1 |
h |
PO, oral; |
DRUGBANK |
Metabolic |
42.0 |
% |
42 |
% |
|
DRUGBANK |
Metabolic |
26.0 |
% |
26 |
% |
|
DRUGBANK |
Metabolic |
16.0 |
% |
16 |
% |
|
DRUGBANK |
Metabolic |
6.0 |
% |
6 |
% |
|
DRUGBANK |
Metabolic |
5.0 |
% |
5 |
% |
|
DRUGBANK |
Metabolic |
5.0 |
% |
5 |
% |
|
DRUGBANK |
Metabolic |
1.0 |
% |
<1 |
% |
|
DRUGBANK |
Clearance |
0.0300 |
L/h/kg |
0.5 |
ml/min/kg |
intravenous injection, IV; human, homo sapiens; |
Human Intravenous Pharmacokinetic Dataset |
Volume of Distribution |
543.0 |
L |
543.0 |
L |
Steady state volume of distribution; |
DRUGBANK |
Volume of Distribution |
3.6 |
L/kg |
3.61 |
L/kg |
intravenous injection, IV; human, homo sapiens; |
Human Intravenous Pharmacokinetic Dataset |
Half-life |
228.0 |
h |
9.5 |
day |
terminal half-life; |
DRUGBANK |
Half-life |
97.0 |
h |
97 |
h |
intravenous injection, IV; human, homo sapiens; |
Human Intravenous Pharmacokinetic Dataset |
Eliminate Route |
62.0 |
% |
62 |
% |
Urinary excretion; |
DRUGBANK |
Eliminate Route |
22.0 |
% |
22 |
% |
Faeces excretion; |
DRUGBANK |
Protein Binding |
99.0 |
% |
99 |
% |
|
DRUGBANK |