Basic Information
Experimental Physicochemical Property
| Property Name | Property Value | Unit | Raw Value | Raw Unit | Reference |
|---|---|---|---|---|---|
| Melting Point | 155.0 | ℃ | 152-158 | ℃ | Product monograph |
Pharmacokinetic/ Toxicokinetic Property
| Property Name | Property Value | Unit | Raw Value | Raw Unit | Annotation | Reference |
|---|---|---|---|---|---|---|
| Absorption | 7.5 | % | 5-10 | % | PO, oral; | DRUGBANK |
| Bioavailability | 1.0 | % | <1 | % | PO, oral; | DRUGBANK |
| T Max | 1.0 | h | 1 | h | PO, oral; | DRUGBANK |
| Half-life | 1.5 | h | ~1.5 | h | elimination half-life; | DRUGBANK |
| Toxicity LD50 | 1531.0 | mg/kg | 1531.0 | mg/kg | PO, oral; mouse; | DRUGBANK | Toxicity LD50 | 1145.0 | mg/kg | 1145.0 | mg/kg | PO, oral; Rattus, Rat; | DRUGBANK | Toxicity LD50 | 154.0 | mg/kg | 154.0 | mg/kg | PO, oral; rabbit; | DRUGBANK |
| Protein Binding | 97.0 | % | 97 | % | plasma proteins; human, homo sapiens; | DRUGBANK |
Maximum Dosage
Not Available
Drug Property Radar Chart
Note: Center: Q1-1.5*IQR, Edge: Q3+1.5*IQR; Q1: Quantile 1, Q3: Quantile 3, IQR: Q3-Q1