Property Name |
Property Value |
Unit |
Raw Value |
Raw Unit |
Annotation |
Reference |
Clearance |
1.9 |
L/h/kg |
31 |
ml/min/kg |
intravenous injection, IV; human, homo sapiens; |
Human Intravenous Pharmacokinetic Dataset |
Volume of Distribution |
4.4 |
L/kg |
4.4 |
L/kg |
intravenous injection, IV; human, homo sapiens; |
Human Intravenous Pharmacokinetic Dataset |
Half-life |
2.2 |
h |
1.7-2.6 |
h |
|
DRUGBANK |
Half-life |
2.6 |
h |
2.6 |
h |
intravenous injection, IV; human, homo sapiens; |
Human Intravenous Pharmacokinetic Dataset |
Toxicity LD50 |
64.0 |
mg/kg |
64.0 |
mg/kg |
intravenous injection, IV; mouse; |
DRUGBANK |
Toxicity LD50 |
540.0 |
mg/kg |
540.0 |
mg/kg |
PO, oral; mouse; |
DRUGBANK |
Toxicity LD50 |
84.0 |
mg/kg |
84.0 |
mg/kg |
intravenous injection, IV; Rattus, Rat; |
DRUGBANK |
Protein Binding |
56.0 |
% |
~56 |
% |
|
DRUGBANK |